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Active pharmaceutical ingredient

Ketotifen Fumarate

Ketotifen Fumarate is a potent antihistamine and mast cell stabilizer commonly used in compounded formulations to manage allergic conditions.

Compounded to order
Prescription required

About this ingredient

Ketotifen fumarate is a salt form of ketotifen, an antihistamine that also has mast cell stabilizing activity.[1] Antihistamines and mast cell stabilizers work together to prevent the release of inflammatory substances from mast cells, reducing allergic responses.[1]

In the United States, ketotifen is available over the counter as an ophthalmic solution containing ketotifen fumarate 0.035% (equivalent to 0.025% ketotifen), labeled to temporarily relieve itchy eyes due to pollen, ragweed, grass, animal hair and dander.[2]

Bayview Pharmacy compounds ketotifen fumarate preparations on a prescriber's order. Compounded ketotifen preparations are not FDA approved.

Compounded at Bayview

How we prepare this ingredient

Patient guides for the preparations we make most often. Each one is compounded to order and requires a prescription.

For prescribers

Full formulary with this ingredient

Every preparation in our formulary that contains this ingredient. Strength, base and dose form are set by the prescription.

Common questions

Frequently asked questions

What is oral ketotifen used for?

Providers may prescribe it off-label as part of a plan for mast cell activation syndrome (MCAS), chronic hives, and other histamine-related conditions. Whether it is appropriate for you is your provider's decision.

Related

Related active ingredients

Other salt forms of this molecule, and ingredients commonly compounded alongside it.

Important information

This page describes an active pharmaceutical ingredient, not a finished drug product. Bayview Pharmacy compounds preparations containing it only on a prescriber's order for an individual patient.

Compounded preparations are not FDA-approved, and the FDA has not evaluated them for safety, effectiveness, or manufacturing quality. Nothing on this page is a claim that any preparation is effective for any condition.

A valid prescription is required. Availability depends on Bayview's licensure in your state. This page is general information, not medical advice — discuss your situation with a licensed healthcare provider.

Talk to a compounding pharmacist

Our pharmacists work with prescribers to build preparations around a patient's dose, form and tolerances. Ask us what is possible with this ingredient.